Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,131
Tocris Bioscience™ TNP-ATP triethylammonium salt
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CAS: 61368-63-6 Molecular Formula: C16H13N8O19P3·C24H64N
| CAS | 61368-63-6 |
|---|---|
| Molecular Formula | C16H13N8O19P3·C24H64N |
2,132
Tocris Bioscience™ KY 02111
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Inhibits canonical Wnt signaling. Promotes differentiation of human ESCs and iPSCs into cardiomyocytes
| CAS | 1118807-13-8 |
|---|---|
| Chemical Name or Material | N-(6-Chloro-2-benzothiazolyl)-3,4-dimethoxybenzenepropanamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C18H17ClN2O3S |
| Formula Weight | Observed MW: 376.86 |
| Assay Percent Range | >99% |
2,133
Tocris Bioscience™ (RS)-(Tetrazol-5-yl)glycine
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Highly potent NMDA agonist
| Target | NMDA Receptor Agonists |
|---|---|
| CAS | 138199-51-6 |
| Solubility | Soluble to 50 mM in water |
| Purity | 98% |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C3H5N5O2 |
| Formula Weight | Observed MW: 143.1 |
| Assay Percent Range | >98% |
2,134
Tocris Bioscience™ Isoguvacine hydrochloride
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CAS: 68547-97-7 Molecular Formula: C6H10ClNO2
| CAS | 68547-97-7 |
|---|---|
| Molecular Formula | C6H10ClNO2 |
2,135
Tocris Bioscience™ Daptomycin
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CAS: 103060-53-3 Molecular Formula: C72H101N17O26
| CAS | 103060-53-3 |
|---|---|
| Molecular Formula | C72H101N17O26 |
2,136
Tocris Bioscience™ RAGE 229
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ctRAGE-DIAPH1 interaction antagonist; reduces inflammatory signaling in diabetic mice
2,137
Tocris Bioscience™ BINA
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CAS: 866823-73-6 Molecular Formula: C30H30O4
| CAS | 866823-73-6 |
|---|---|
| Molecular Formula | C30H30O4 |
2,138
Tocris Bioscience™ AMG 510
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Potent and selective KRASG12C inhibitor
| Target | Ras GTPase Inhibitors |
|---|---|
| CAS | 2252403-56-6 |
| Purity | 0.98 |
| Chemical Name or Material | (1 R)-6-Fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-[4-methyl-2-(1-methylethyl)-3-pyridinyl]-4-[(2 S)-2-methyl-4-(1-oxo-2-propen-1-yl)-1-piperazinyl]pyrido[2,3-d]pyrimidin-2(1 H)-one |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C30H30F2N6O3 |
2,139
Tocris Bioscience™ BMS 566419
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Inosine monophosphatase dehydrogenase (IMPDH) inhibitor
| Target | Dehydrogenase Inhibitors |
|---|---|
| CAS | 566161-24-8 |
| Purity | >98% |
| Chemical Name or Material | N-[1-[6-(4-Ethyl-1-piperazinyl)-3-pyridinyl]-1-methylethyl]-2-fluoro-9,10-dihydro-9-oxo-3-acridinecarboxamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C28H30FN5O2 |
| Formula Weight | 487.57 |
2,140
Tocris Bioscience™ S 24795
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CAS: 304679-75-2 Molecular Formula: C14H13BrINO
| CAS | 304679-75-2 |
|---|---|
| Molecular Formula | C14H13BrINO |
2,141
Tocris Bioscience™ PF 04620110
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Potent and selective DGAT-1 inhibitor; orally bioavailable
| CAS | 1109276-89-2 |
|---|---|
| Chemical Name or Material | trans-4-[4-(4-Amino-7,8-dihydro-5-oxopyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl]cyclohexaneacetic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C21H24N4O4 |
| Formula Weight | Observed MW: 396.44 |
| Assay Percent Range | >98% |
2,142
Tocris Bioscience™ DZNep HCl
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3-Deazaneplanocin A hydrochloride synthesized to Ancillary Material Grade
2,143
Tocris Bioscience™ PPY A
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CAS: 875634-01-8 Molecular Formula: C22H20N4O2
| CAS | 875634-01-8 |
|---|---|
| Molecular Formula | C22H20N4O2 |
2,144
Tocris Bioscience™ AM 6545
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High affinity and selective CB1 antagonist
| CAS | 1245626-05-4 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 20mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | AM 6545 |
| Recommended Storage | Store at 4°C |
| Synonym | 5-[4-(4-Cyano-1-butyn-1-yl)phenyl]-1-(2,4-dichlorophenyl)-N-(1,1-dioxido-4-thiomorpholinyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Molecular Formula | C26H23Cl2N5O3S |
| Formula Weight | 556.46 |
2,145
Tocris Bioscience™ GNF 5
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CAS: 778277-15-9 Molecular Formula: C20H17F3N4O3
| CAS | 778277-15-9 |
|---|---|
| Molecular Formula | C20H17F3N4O3 |